Publication Beamlines Strategic Pillar
Gunn, R.J.; Lawson, J.D.; Ivetac, A.; Ulaganathan, T.; Coulombe, R. et al. (2024). SOS2 crystal structure with fragment bound (compound 13). Protein Data Bank: 8t5r. CMCF-BM Agriculture
Smith, Christopher R.; Chen, Dan; Christensen, James G.; Coulombe, René; Féthière, James et al. (2023). Discovery of Five SOS2 Fragment Hits with Binding Modes Determined by SOS2 X-Ray Cocrystallography. Journal of Medicinal Chemistry 67(1) , 774-781. 10.1021/acs.jmedchem.3c02140. [PDB: 8t5g, 8t5m, 8t5r] CMCF-BM, CMCF-ID Health
Li, K.; Tokareva, O.S.; Thomson, T.M.; Verdine, G.L.; McGee, J.H. et al. (2023). Crystal structure of the WWP1 HECT domain in complex with H302, a Helicon Polypeptide. Protein Data Bank: 8ei4. CMCF-BM Agriculture
Musil, D.; Toure, M. (2023). CRYSTAL STRUCTURE OF HUMAN HPK1 (MAP4K1) COMPLEX WITH 2-[8-Amino-7-fluoro-6-(8-methyl-2,3-dihydro-1H-pyrido[2,3-b][1,4]oxazin-7-yl)-isoquinolin-3-ylamino]-6-isopropyl-5,6-dihydro-4H-1,6,8a-triaza-azulen-7-one. Protein Data Bank: 8cij. CMCF-BM Agriculture
Toure, Momar; Johnson, Theresa; Li, Bin; Schmidt, Ralf; Ma, Hong et al. (2023). Discovery of quinazoline HPK1 inhibitors with high cellular potency. Bioorganic and Medicinal Chemistry 92, 117423. 10.1016/j.bmc.2023.117423. [PDB: 8cij] CMCF-BM Health
Bian, M.J.; Cheng, Q.P.; Wang, P.; Zhu, G.P. (2023). Crystal structure of isocitrate dehydrogenase from Campylobacter corcagiensis. Protein Data Bank: 7y1u. CMCF-BM Health
Gui, Wenjun; Hang, Yumo; Cheng, Wang; Gao, Minqi; Wu, Jiaquan et al. (2023). Structural basis of CDK3 activation by cyclin E1 and inhibition by dinaciclib. Biochemical and Biophysical Research Communications 662, 126-134. 10.1016/j.bbrc.2023.04.026. CMCF-BM, CMCF-ID Health
Li, K.; Callahan, A.J.; Travaline, T.L.; Tokareva, O.S.; Swiecicki, J.-M. et al. (2023). Structure of the STUB1 TPR domain in complex with H204, an all-D Helicon Polypeptide. Protein Data Bank: 8f17. CMCF-BM Agriculture
Li, K.; Callahan, A.J.; Travaline, T.L.; Tokareva, O.S.; Swiecicki, J.-M. et al. (2023). Structure of the STUB1 TPR domain in complex with H203, an all-D Helicon Polypeptide. Protein Data Bank: 8f16. CMCF-BM Agriculture
Callahan, Alex J.; Gandhesiri, Satish; Travaline, Tara L.; Lozano Salazar, Lia; Hanna, Stephanie et al. (2023). Single-Shot Flow Synthesis of D-Proteins for Mirror-Image Phage Display. Environmental Science & Technology . 10.26434/chemrxiv-2023-x86xp. [PDB: 8f16, 8f17] CMCF-BM Health
Ghosh, K. (2024). Human CK1 Delta Kinase structure bound to Inhibitor. Protein Data Bank: 8izc. CMCF-ID Health
Perez-Bermejo, Juan A.; Efagene, Oghene; Matern, William M.; Holden, Jeffrey K.; Kabir, Shaheen et al. (2024). Functional screening in human HSPCs identifies optimized protein-based enhancers of Homology Directed Repair. Nature Communications 15(1) . 10.1038/s41467-024-46816-5. [PDB: 8svg, 8svh, 8svi] CMCF-ID Health
Partridge, J.R.; Holden, J.K.; Wibowo, A.S.; Mulichak, A. (2024). Ubiquitin variant i53:Mutant L67H with 53BP1 Tudor domain. Protein Data Bank: 8svi. CMCF-ID Agriculture
Holden, J.K.; Partridge, J.R.; Wibowo, A.S.; Mulichak, A. (2024). Ubiquitin variant i53 mutant L67R bound to 53BP1 Tudor Domain. Protein Data Bank: 8svh. CMCF-ID Agriculture
Holden, J.K.; Partridge, J.R.; Wibowo, A.S.; Mulichak, A. (2024). Ubiquitin variant i53 in complex with 53BP1 Tudor domain. Protein Data Bank: 8svg. CMCF-ID Agriculture